Hair GrowthSkin HealthNo data

Acetyl Tetrapeptide-3

Acetyl Tetrapeptide-3

Overview

Acetyl Tetrapeptide-3 is a synthetic biomimetic tetrapeptide that stimulates extracellular matrix proteins in the scalp and promotes hair follicle anchoring and growth. It is primarily used as a cosmetic ingredient in anti-hair loss formulations and has shown clinical efficacy in reducing hair loss and improving hair density in controlled studies. Unlike hormonal approaches to hair loss Acetyl Tetrapeptide-3 works by strengthening the structural support of the hair follicle in the scalp making it particularly useful for diffuse thinning and age-related hair loss where follicle miniaturization is the primary mechanism.

Mechanism of Action

Acetyl Tetrapeptide-3 mimics the signal peptides involved in extracellular matrix remodeling around hair follicles. It stimulates the synthesis of laminin-5 and collagen IV in the dermal papilla and basement membrane — structural proteins that anchor hair follicles in the scalp and maintain their integrity. By reinforcing the follicle anchoring structure Acetyl Tetrapeptide-3 reduces hair shedding and extends the anagen growth phase. It also activates stem cell niches in the hair follicle bulge region promoting the differentiation of progenitor cells into new hair matrix cells. Clinical studies have demonstrated significant reductions in hair loss measured by phototrichogram and improvements in hair density and thickness comparable to minoxidil-containing formulations when used at effective concentrations.

Where does Acetyl Tetrapeptide-3 sit?

See how this peptide compares across all 85 peptides in our database.

Dosage Information

Typical Dose

500 ppm (0.05%) in topical formulation

Frequency

Twice daily application to affected areas

Administration

Topical serum or lotion

Notes

Most clinical evidence uses concentrations of 500-3000 ppm. Often combined with other hair peptides like biotinoyl tripeptide-1 for synergistic effects. Results typically visible after 3-4 months of consistent use.

Compound Data

Acetyl Tetrapeptide-3 structure

Molecular Formula

C22H39N9O5

Molecular Weight

509.60 g/mol

IUPAC Name

(2S)-2-[[(2S)-2-[[2-[[(2S)-2-acetamido-6-aminohexanoyl]amino]acetyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-6-aminohexanamide

PubChem CID

11752568

Potential Side Effects

Very well tolerated in clinical studiesScalp irritation in sensitive individuals (rare)Contact allergy (very rare)

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Quick Facts

Administration
Topical serum or lotion
Typical Dose
500 ppm (0.05%) in topical formulation
Frequency
Twice daily application to affected areas
References
0 curated + 1 from PubMed
Evidence Score
12.3 / 100