Skin HealthAnti-AgingEmergingHuman trials

Syn-Coll

Palmitoyl Tripeptide-5

Overview

Syn-Coll (Palmitoyl Tripeptide-5) is a synthetic lipopeptide that mimics the natural activation mechanism of TGF-β — the primary growth factor responsible for collagen synthesis in the skin. Unlike GHK-based peptides that stimulate collagen indirectly through matrikine signaling Syn-Coll directly activates the TGF-β receptor pathway producing a more targeted collagen synthesis stimulus. It has demonstrated significant improvements in skin firmness and wrinkle reduction in clinical trials and is used in prestige anti-aging skincare formulations.

Mechanism of Action

Palmitoyl Tripeptide-5 mimics the sequence Lys-Arg-Phe-Lys from thrombospondin-1 — a naturally occurring activator of latent TGF-β. By binding to the same thrombospondin-1 receptor site on latent TGF-β this peptide triggers the conformational change that activates TGF-β releasing it from its inactive latent complex. Active TGF-β then binds to TGF-β receptors on fibroblasts activating the SMAD signaling cascade that upregulates transcription of collagen types I and III elastin and other extracellular matrix components. This direct TGF-β activation mechanism is more targeted than matrikine-based approaches and produces a strong collagen synthesis response in clinical studies.

Dosage Information

Typical Dose

4-8% concentration in topical formulation

Frequency

Once or twice daily

Administration

Topical serum or cream

Notes

Effective as a standalone anti-aging ingredient but also works synergistically with Matrixyl 3000 (Palmitoyl Tripeptide-1 + Palmitoyl Tetrapeptide-7) for comprehensive collagen support.

Where does Syn-Coll sit?

See how this peptide compares across all 111 peptides in our database.

Evidence Score

0.55

Clinical trials
0.8335%
Literature
0.3430%
Community
0.0020%
Completeness
1.0015%
1 clinical trials1 reviews

Compound Data

Syn-Coll structure

Molecular Formula

C33H65N5O5

Molecular Weight

611.90 g/mol

IUPAC Name

(2S)-6-amino-2-[[(2S)-2-[[(2S)-6-amino-2-(hexadecanoylamino)hexanoyl]amino]-3-methylbutanoyl]amino]hexanoic acid

PubChem CID

11950477

Potential Side Effects

Well tolerated in clinical studiesMild skin sensitivity in very reactive skin (rare)No known systemic effects

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Quick Facts

Administration
Topical serum or cream
Typical Dose
4-8% concentration in topical formulation
Frequency
Once or twice daily
References
0 curated + 3 from PubMed
Clinical Trials
2 registered
Evidence Score
0.5 / 100